Endocrine & Hormonal Agents – Antidiabetic, Hormonal Supplements, Contraceptives & HRT

Introduction

Endocrine and hormonal therapies are essential in the management of diabetes, thyroid disorders, adrenal insufficiency, reproductive health, and menopause. Nirvana Pharma provides a comprehensive portfolio covering oral antidiabetic agents, insulin preparations, hormonal supplements, contraceptives, and hormone replacement therapies to support diverse patient needs.


🔹 Antidiabetic Agents

A. Biguanides

Drug Strengths Notes
Metformin 500, 850, 1000 mg; ER: 500, 750, 1000 mg First-line in T2DM

B. Sulfonylureas

Drug Strengths Notes
Glimepiride 1, 2, 4 mg Once daily
Glyburide (Glibenclamide) 2.5, 5 mg
Glipizide 5, 10 mg; ER: 2.5–10 mg

C. Meglitinides (Glinides)

Drug Strengths Notes
Repaglinide 0.5, 1, 2 mg Pre-meal dosing
Nateglinide 60, 120 mg

D. Thiazolidinediones (TZDs)

Drug Strengths Notes
Pioglitazone 15, 30, 45 mg Improves insulin sensitivity

E. DPP-4 Inhibitors

Drug Strengths Notes
Sitagliptin 25, 50, 100 mg Oral, well tolerated
Vildagliptin 50 mg
Linagliptin 5 mg

F. SGLT-2 Inhibitors

Block glucose reabsorption in the kidney → lower blood sugar, promote weight loss, reduce CV and renal risk.

Drug Strengths Notes
Dapagliflozin 5 mg, 10 mg CV + renal benefits
Empagliflozin 10 mg, 25 mg Strong CV outcome data
Canagliflozin 100 mg, 300 mg CV + renal benefits; monitor for amputation risk
Ertugliflozin (Steglatro®) 5 mg, 15 mg Initial: 5 mg once daily; may increase to 15 mg after 4–12 weeks; Max: 15 mg/day

G. GLP-1 Receptor Agonists

Injectable Agents

Drug Dosing Frequency Common Strengths Key Notes
Exenatide SC twice daily 5 mcg, 10 mcg First GLP-1 agonist; short-acting
Exenatide ER SC once weekly 2 mg Extended-release, more convenient
Lixisenatide (not available in US/Canada) SC once daily 10 mcg, 20 mcg Short-acting, used with basal insulin
Liraglutide SC once daily 0.6 mg, 1.2 mg, 1.8 mg CV benefit, weight loss, widely used
Dulaglutide SC once weekly 0.75 mg, 1.5 mg, 3 mg, 4.5 mg Weekly dosing, good tolerability
Semaglutide (inj.) SC once weekly 0.25 mg, 0.5 mg, 1 mg, 2 mg High efficacy for weight loss & CV outcomes
Tirzepatide (dual GIP/GLP-1 agonist) SC once weekly 2.5 mg, 5 mg, 7.5 mg, 10 mg, 12.5 mg, 15 mg Dual incretin effect, superior HbA1c & weight loss outcomes

Oral Agents

Drug Dosing Frequency Common Strengths Key Notes
Semaglutide (Rybelsus®) Oral, once daily 3 mg, 7 mg, 14 mg First oral GLP-1 agonist, requires fasting administration
Oral formulations (under study) (e.g., R2 variants) 1.5 mg, 4 mg, 9 mg Investigational strengths

🔹 Insulin Therapy

Type Examples Strengths
Rapid-acting Lispro, Aspart, Glulisine 100 U/mL pens/vials
Short-acting Regular Insulin 100 U/mL vials
Intermediate NPH 100 U/mL
Long-acting Glargine, Detemir, Degludec 100–200 U/mL

🔹 Thyroid Hormones

Drug Strengths Notes
Levothyroxine (T4) 25–150 mcg Hypothyroidism
Liothyronine (T3) 5, 25 mcg Rapid onset
T4 + T3 combo Various Rarely used

🔹 Corticosteroids

Drug Strengths Notes
Prednisone 5, 10, 20 mg Oral anti-inflammatory
Prednisolone 5, 10 mg tab; Syrup: 15 mg/5 mL Pediatric common
Methylprednisolone 4, 8, 16 mg; Inj: 40, 125 mg
Dexamethasone 0.5, 4 mg tab; Inj: 4 mg/mL Potent, long-acting
Hydrocortisone 10, 20 mg tab; Inj: 100 mg vials Replacement, acute

🔹 Contraceptives & HRT

A. Oral Contraceptives (Combined Estrogen + Progestin)

Components Common Strengths
EE + Levonorgestrel EE 30 mcg + LNG 150 mcg
EE + Drospirenone EE 30 mcg + DRSP 3 mg
EE + Desogestrel EE 30 mcg + DSG 150 mcg
EE + Norethindrone EE 20–35 mcg + NETA 1 mg

B. Progestin-only Contraceptives

Drug Strengths
Norethindrone 0.35 mg daily
Desogestrel 75 mcg daily
Levonorgestrel (IUD/implant) IUD: 52 mg (5 yrs), Implant: 68 mg (3 yrs)

C. Emergency Contraceptives

Drug Strengths
Levonorgestrel 1.5 mg single dose
Ulipristal acetate 30 mg single dose

D. Hormone Replacement Therapy (HRT)

Drug / Combo Strengths
Estradiol (oral/patch/gel) Tab: 1–2 mg; Patch: 0.025–0.1 mg/day
Conjugated estrogens Tab: 0.3, 0.625, 1.25 mg
Estradiol + Progesterone Various combos (e.g., E2 1 mg + Prog 100 mg)
Medroxyprogesterone acetate 2.5, 5, 10 mg

Closing Note

With a broad endocrine and hormonal therapy portfolio, Nirvana Pharma addresses the complete spectrum of diabetes care, hormone replacement, contraceptive options, and steroid therapy—backed by quality formulations trusted in clinical practice.

Add to cart